I-BET282 ts-2 Thr-Thr-Tyr-Ala-Asp-Phe-Ile-Ala-Ser-Gly-Arg-Thr-Gly-Arg-Arg-Asn-Ala-Ile-His-Asp

Thr-Thr-Tyr-Ala-Asp-Phe-Ile-Ala-Ser-Gly-Arg-Thr-Gly-Arg-Arg-Asn-Ala-Ile-His-Asp

Solubility: DMSO : 250 mg/mL (813

Loganin attenuates H2O2-induced neuronal damage via suppressing MAPKs signals in SH-SY5Y cells[2]

In one of the experiments

modulating non-selective cation channels (NSC)

I-BET282 ts-2 Thr-Thr-Tyr-Ala-Asp-Phe-Ile-Ala-Ser-Gly-Arg-Thr-Gly-Arg-Arg-Asn-Ala-Ile-His-AspI BET282 is a pan inhibitor of all eight BET bromodomains, and selectivity over other representative bromodomain containing proteins. I BET282 shows pIC50s ranging 6. 4 7. 7 for BRD2 (BD1 BD2), BRD2 (BD1 BD), BRD3 (BD1 BD), and BRD4 (BD1 BD). Product information CAS Number: 1422554 34 4 Molecular Weight: 450. 53 Formula: C25H30N4O4 Chemical Name: 4 {8 methoxy 1 [(2R) 1 methoxypropan 2 yl] 2 (oxan 4 yl) 1H imidazo[4,5 c]quinolin 7 yl} 3,5 dimethyl 1,2