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InChiKey: JRNWTJUIMRLKBV-UHFFFAOYSA-N
It is a weak inhibitor of PKA with an IC50 of 30 μM
Smiles: COC1=CC(=CC=C1NC1=CC(NC2=CC=CC=C2C(=O)NC)=C(C=N1)C(F)(F)F)N1CCOCC1
NS11394 is unique in having superior efficacy at GABA(A)-alpha(3) receptors while maintaining low efficacy at GABA(A)-alpha(1) receptors
It may also inhibit the synthesis of spermidine in mycobacteria
EN4 MYC inhibitor - CAS# 1197824-15-9 degrader-1 InChiKey: JRNWTJUIMRLKBV-UHFFFAOYSA-NEN4 is a functional Covalent Ligand Targeting an Intrinsically Disordered Cysteine within MYC. EN4 functionally and covalently targets an intrinsically disordered region in MYC. EN4 directly targets MYC in cells and reduces MYC and MAX thermal stability. EN4 inhibits MYC activity, downregulates MYC targets, and impairs tumorigenesis. MYC is a major oncogenic transcriptional driver of most human cancers that has remained intractable to direct targeting
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